Gabapentinoids: Difference between revisions

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m Added Baclofen as an example.
>Discount Pharmacologist
alternative name
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[[File:Gabapentinoidsstructure.png|250px|thumbnail|Diagram showing the structural similarities of [[GABA|gamma-aminobutyric acid]] (GABA), [[pregabalin]] and [[gabapentin]].]]
[[File:Gabapentinoidsstructure.png|250px|thumbnail|Diagram showing the structural similarities of [[GABA|gamma-aminobutyric acid]] (GABA), [[pregabalin]] and [[gabapentin]].]]


'''Gabapentinoids''' are a relatively small chemical class of [[psychoactive substances]] derived from [[GABA|gamma-aminobutyric acid]] (GABA).{{citation needed}} Members of this class include [[gabapentin]], [[F-phenibut]], [[phenibut]] and [[pregabalin]].  
'''Gabapentinoids''', also known as α<sub>2</sub>δ ligands, are a relatively small chemical class of [[psychoactive substances]] derived from [[GABA|gamma-aminobutyric acid]] (GABA).{{citation needed}} Members of this class include [[gabapentin]], [[F-phenibut]], [[phenibut]] and [[pregabalin]].  


Gabapentinoids are commonly prescribed for epilepsy, neuropathic pain, and [[restless legs syndrome]]. [[Subjective effects]] include [[sedation]], [[muscle relaxation]], and [[anxiety suppression]].  
Gabapentinoids are commonly prescribed for epilepsy, neuropathic pain, and [[restless legs syndrome]]. [[Subjective effects]] include [[sedation]], [[muscle relaxation]], and [[anxiety suppression]].  
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==Examples==
==Examples==
*[[F-Phenibut]]
*[[F-Phenibut]]
*[[Gabapentin]]
*[[Gabapentin]]
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==See also==
==See also==
*[[Responsible use]]
*[[Responsible use]]
*[[Depressants]]
*[[Depressants]]
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==External links==
==External links==
*[https://en.wikipedia.org/wiki/Gabapentinoid Gabapentinoid (Wikipedia)]
*[https://en.wikipedia.org/wiki/Gabapentinoid Gabapentinoid (Wikipedia)]


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[[Category:Chemical class]]
[[Category:Chemical class]]
[[Category:Pharmacology]]
[[Category:Pharmacology]]
<references />