Talk:Troparil: Difference between revisions

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+{{headerpanel|{{Approval}}{{stub}}}}
+{{SummarySheet}}
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 {{SubstanceBox/Troparil}}
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 ==Pharmacology==
-{| class="wikitable" style="float:right"
+Troparil primarily acts as a dopamine [[reuptake inhibitor]] (DRI). While this effect is a few times more potent as with cocaine, the effect of troparil on serotonin reuptake inhibition is slightly less pronounced.
-|+ Binding profile of troparil compared to cocaine
-! || colspan="3"| IC<sub>50</sub> (nM)
-|-
-! Compound !! DAT !! NET !! SERT
-|-
-| Troparil || 23 ± 5 || 920 ± 73 || 1962 ± 61
-|-
-| Cocaine || 89 ± 4.8 || 3298 ± 293 || 1045 ± 89
-|}
-Troparil primarily acts as a dopamine [[reuptake inhibitor]] (DRI). While this effect is a few times more potent as with cocaine, the effect of troparil on serotonin reuptake inhibition is slightly less pronounced.<ref>Cocaine and 3.beta.-(4'-Substituted phenyl)tropane-2.beta.-carboxylic Acid Ester and Amide Analogs. New High-Affinity and Selective Compounds for the Dopamine Transporter | http://pubs.acs.org/doi/abs/10.1021/jm00002a020</ref>
+{{Binding profiles of tropane stimulants}}
 ==Subjective effects==
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 *[[Responsible use]]
 ==External links==
+*[[wikipedia:Troparil|Troparil (Wikipedia)]]
+*[https://isomerdesign.com/PiHKAL/explore.php?id=2977 Troparil (Isomer Design)]
 ==Literature==
 ==References==
 <references />
-[[Category:Psychoactive substance]][[Category:Tropane]][[Category:Stimulant]][[Category:Research chemical]][[Category:Proofread]][[Category:Approval]]
+[[Category:Psychoactive substance]]
+[[Category:Phenyltropane]]
+[[Category:Stimulant]]
+[[Category:Research chemical]]
+[[Category:Proofread]]
+[[Category:Approval]]